Tirzepatide ingano, mbiri-inobata glucose-inotsamira insulinotropic polypeptide (GIP) uye glucagon-yakafanana peptide-1 (GLP-1) receptor agonist. Inomiririra kufambira mberi kwakakosha mukurapa kwechirwere cheshuga 2 uye yakaratidza mhedzisiro inovimbisa mukutonga uremu. Tirzepatide jekiseni poda ndiyo fomu yemishonga inoshandiswa kugadzirira mhinduro ye subcutaneous administration.
Nzira Yekuita
Tirzepatide inoshanda nekuita zvese zviri zviviri GIP uye GLP-1 receptors, izvo zvinosanganisirwa mukudzora mazinga eshuga yeropa uye kudya. Iyo mbiri agonism inopa akati wandei maitiro anobatsira:
Enhanced Insulin Secretion: Inokurudzira kusunungurwa kwe insulini nenzira inotsamira shuga, zvichibatsira kuderedza mazinga eshuga yeropa pasina kukonzera hypoglycemia.
Yakadzvanywa Glucagon Release: Inoderedza secretion yeglucagon, hormone inosimudza mazinga eshuga.
Appetite Regulation: Inosimudzira satiety uye inoderedza kudya kwekudya, zvichiita kuti uremu huremerwe.
Yakanonoka Gastric Emptying: Inononoka kubuda mudumbu, iyo inobatsira mukudzora postpandial shuga yeropa.
Kushandiswa Kwakabvumirwa
Nezvezvichangoburwa, Tirzepatide yakatenderwa nezviremera zvinodzora zvakaita seUS Food and Drug Administration (FDA) yekurapa chirwere cheshuga cherudzi rwechipiri. Iri zvakare pasi pekuferefetwa nekuda kwekushandisa kwayo mukugadzirisa kufutisa.
Benefits
Inoshanda Glycemic Kudzora: Kudzikira kwakakosha mumazinga eHbA1c.
Kurasikirwa Kwehuremu: Kuderedza uremu, izvo zvinobatsira kune varwere vane Type 2 chirwere cheshuga uye kufutisa.
Cardiovascular Benefits: Inogona kuvandudzwa muhutano hwemoyo ngozi zvinhu, kunyange zvazvo zvidzidzo zvinoenderera mberi zviri kuwedzera kuongorora chinhu ichi.
Kusununguka: Kamwe-vhiki nevhiki dosing inovandudza kutevedzera kwevarwere kana ichienzaniswa nemishonga yemazuva ese.
Zvingangoitika Zvikonzero
Nepo Tirzepatide ichiwanzo bvumidzwa, vamwe vashandisi vanogona kusangana nemhedzisiro, kusanganisira:
Matambudziko eGastrointestinal:
Nausea, kurutsa, manyoka, uye kusvotekana zvinowanzoitika, kunyanya panguva yekutanga kurapwa.
Ngozi yeHypoglycemia: Kunyanya kana yakashandiswa pamwe chete nemimwe mishonga inoderedza shuga.
Pancreatitis: Kashoma asi yakakomba, inoda kurapwa nekukurumidza kana zviratidzo zvakaita sekurwadziwa kwakanyanya mudumbu zvikaitika.
Kugadzirira uye Kutungamirira
Tirzepatide jekiseni poda inoda kudzokororwa nemushonga wakakodzera (unowanzo kupihwa mukiti) kugadzira mhinduro yejekiseni. Mhinduro yakagadziridzwa inofanira kuva yakajeka uye isina zvimedu. Inoitwa pasi pasi mudumbu, chidya, kana kumusoro ruoko.