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Glucagon

Tsanangudzo Pfupi

Glucagon ndeye yakasikwa peptide hormone inoshandiswa sechimbichimbi kurapwa kune yakanyanya hypoglycemia uye yakaverengerwa basa rayo mukugadzirisa metabolic, kuonda, uye digestive diagnostics.


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Glucagon API

Glucagon ndeye yakasikwa peptide hormone inoshandiswa sechimbichimbi kurapwa kune yakanyanya hypoglycemia uye yakaverengerwa basa rayo mukugadzirisa metabolic, kuonda, uye digestive diagnostics.

 

Mechanism & Tsvagiridzo:

Glucagon inosunga kune glucagon receptor (GCGR) muchiropa, ichikurudzira:

Glycogen kuputsika kuwedzera shuga yeropa

Lipolysis uye kuunganidza simba

Gastrointestinal motility modulation (inoshandiswa muradiology)

Iri zvakare kuongororwa mukufutisa, mhando 2 chirwere cheshuga, uye maviri / katatu agonist ekurapa neGLP-1 uye GIP.

 

API Zvimiro (Gentolex Boka):

Yakakwirira-kuchena peptide (≥99%)

Yakagadzirwa kuburikidza ne-soli-phase peptide synthesis (SPPS)

GMP-yakafanana nemhando

Inokodzera majekiseni nemakiti ekukurumidzira

Glucagon API yakakosha pakununura hypoglycemia, diagnostic imaging, uye metabolic disorder research.


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