Products
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High Purity Peptides Retatrutide 10mg yeKurasikirwa Kwehuremu uye Chirwere cheshuga
Kuchena:> 99%
Nyika: Lyophilized Powder
Kuonekwa: White powder
Tsanangudzo: 5mg/10mg/15mg/20mg/30mg
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Retatrutide
Retaglutide itsva dipeptidyl peptidase-4 (DPP-4) inhibitor class hypoglycemic drug inogona kudzivirira kuparara kweglucagon-like peptide-1 (GLP-1) uye glucose-inotenderera insulin-releasing polypeptide (GIP) neDPP-4 enzyme mumatumbo uye ropa, nekuwedzera pancreatic masero, kuwedzera pancreatic masero. basal level yekutsanya insulin, nepo ichideredza secretion yeglucagon nepancreatic α masero, nekudaro zvakanyanya kunyatso kudzora postprandial shuga yeropa. Inoita zvakanaka maererano neiyo hypoglycemic effect, kushivirira, uye kutevedzera.
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Inclisiran sodium
Inclisiran sodium API (Active Pharmaceutical Ingredient) inodzidzwa kunyanya mumunda weRNA kupindira (RNAi) uye kurapa kwemwoyo. SeSiRNA ine tambo mbiri yakanangana nePCSK9 gene, inoshandiswa mu preclinical uye kiriniki yekutsvagisa kuongorora maitiro-akareba-anoita gene-kunyarara nzira dzekudzikisa LDL-C (yakaderera-density lipoprotein cholesterol). Iyo inoshandawo semuenzaniso wekomboni yekuongorora siRNA yekuendesa masisitimu, kugadzikana, uye chiropa-yakanangwa RNA therapeutics.
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Fmoc-Gly-Gly-OH
Fmoc-Gly-Gly-OH idipeptide inoshandiswa sechinhu chekutanga chekuvaka mune yakasimba-phase peptide synthesis (SPPS). Iyo inoratidzira maviri glycine zvakasara uye Fmoc-yakachengetedzwa N-terminus, inobvumira inodzorwa peptide cheni kureba. Nekuda kwehukuru hudiki hweglycine uye kuchinjika, dipeptide iyi inowanzodzidzwa mukati meiyo peptide backbone dynamics, linker dhizaini, uye chimiro chekumisikidza mumapeptide nemapuroteni.
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Fmoc-Thr(tBu)-Phe-OH
Fmoc-Thr(tBu)-Phe-OH idipeptide building block inowanzoshandiswa mune yakasimba-phase peptide synthesis (SPPS). Fmoc (9-fluorenylmethyloxycarbonyl) boka rinodzivirira N-terminus, nepo tBu (tert-butyl) boka rinodzivirira hydroxyl side chain yethreonine. Iyi dipeptide yakadzivirirwa inodzidzwa nezve basa rayo mukufambisa kwakaringana peptide kurebesa, kudzikisira kumhanya, uye kuenzanisira chaiyo inoteedzana modhi muchimiro cheprotein uye zvidzidzo zvekudyidzana.
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AEEA-AEEA
AEEA-AEEA is hydrophilic, inochinjika spacer inowanzoshandiswa mu peptide uye zvinodhaka conjugation research. Inosanganisira maviri ethylene glycol-based units, zvichiita kuti zvive zvakakosha pakudzidza migumisiro ye linker kureba uye kushanduka pakubatana kwema molecular, solubility, uye biological chiitiko. Vatsvagiri vanowanzo shandisa zvikamu zveAEEA kuongorora kuti ma spacers anopesvedzera sei mashandiro eantibody-drug conjugates (ADCs), peptide-drug conjugates, uye mamwe bioconjugates.
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Fmoc-L-Lys[Eic(OtBu)-γ-Glu(OtBu)-AEEA]-OH
Mushonga uyu unodzivirirwa, unoshanda lysine derivative inoshandiswa mu peptide synthesis uye drug conjugate development. Inosanganisira Fmoc boka reN-terminal kudzivirira, uye rutivi-cheni kuchinjwa neEic (OtBu) (eicosanoic acid derivative), γ-glutamic acid (γ-Glu), uye AEEA (aminoethoxyethoxyacetate). Izvi zvikamu zvakagadzirirwa kudzidza lipidation mhedzisiro, spacer chemistry, uye inodzorwa kuburitswa kwezvinodhaka. Inotsvakurudzwa zvakanyanya mumamiriro ezvinhu emishonga yeprodrug, ADC linkers, uye membrane-interacting peptides.
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Fmoc-L-Lys[Ste(OtBu)-γ-Glu-(OtBu)-AEEA-AEEA]-OH
Mushonga uyu wakagadziridzwa lysine derivative inoshandiswa mupeptide synthesis, kunyanya pakuvaka anonangwa kana akawanda anoshanda peptide conjugates. Boka reFmoc rinobvumira nhanho synthesis kuburikidza neFmoc solid-phase peptide synthesis (SPPS). Cheni yepadivi yakagadziridzwa ine stearic acid inotorwa (Ste), γ-glutamic acid (γ-Glu), uye maviri AEEA (aminoethoxyethoxyacetate) linkers, ayo anopa hydrophobicity, kuchaja zvivakwa, uye kuchinjika nzvimbo. Inowanzodzidzwa nezvebasa rayo muhurongwa hwekuunza zvinodhaka, kusanganisira antibody-drug conjugates (ADCs) uye cell-inopinda peptides.
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Liraglutide Anti-Diabetics yeRopa Shuga Kudzora CAS NO.204656-20-2
Active Ingredient:Liraglutide (analog yemunhu glucagon-like peptide-1 (GLP-1) inogadzirwa nembiriso kuburikidza neiyo genetic recombination tekinoroji).
Chemical Name:Arg34Ls26-(N-e-(γ-Glu(N-α-hexadecanoyl)))-GLP-1[7-37]
Zvimwe Ingredients:Disodium Hydrogen Phosphate Dihydrate, Propylene Glycol, Hydrochloric Acid uye/kana Sodium Hydroxide (se pH Adjusters Chete), Phenol, uye Mvura Yejekiseni.
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Leuprorelin Acetate Inogadzirisa Secretion yeGonadal Hormones
Zita: Leuprorelin
Nhamba yeCAS: 53714-56-0
Molecular formula: C59H84N16O12
Molecular uremu: 1209.4
Nhamba yeEINECS: 633-395-9
Kutenderera chaiko: D25 -31.7° (c = 1 mu1% acetic acid)
Density: 1.44±0.1 g/cm3(Zvakafanotaurwa)
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Boc-His(Trt)-Aib-Gln(Trt)-Gly-OH
Boc-His(Trt)-Aib-Gln(Trt)-Gly-OHtetrapeptide yakachengetedzwa inoshandiswa mu peptide synthesis uye zvidzidzo zvemaitiro. Boka reBoc (tert-butyloxycarbonyl) rinodzivirira N-terminus, nepo Trt (trityl) mapoka anodzivirira cheni dzeparutivi dze histidine uye glutamine kudzivirira kuita kusingadiwe. Kuvapo kweAib (α-aminoisobutyric acid) kunokurudzira kuumbwa kwehelical uye kunowedzera kugadzikana kwepeptide. Iyi peptide yakakosha pakuongorora kupeta peptide, kugadzikana, uye sechikafu chekugadzira biologically active peptides.
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BPC-157
BPC-157 API inoshandisa solid phase synthesis (SPPS) maitiro:
Kuchena kwepamusoro: ≥99% (HPLC kuonekwa)
Yakaderera tsvina yakasara, hapana endotoxin, hapana inorema simbi kusvibiswa
Batch kugadzikana, kudzokorora kwakasimba, kutsigira jekiseni nhanho kushandiswa
Tsigira giremu uye kilogiramu nhanho yekupa kuti isangane nezvinodiwa zvematanho akasiyana kubva kuR&D kusvika kumaindasitiri.
