Zita | Sildenafil Citrate |
Nhamba | 171599-83-0 |
Molecular Formula | C28h38n6o11s |
Sreek inoremerwa | 666.70 |
Einecs nhamba | 200-659-6 |
Merck | 14,8489 |
Density | 1.445G / cm3 |
Kuchengetedza mamiriro | 2-8 ° C |
Fomu | Poda |
Ruvara | Chena |
Solubility yemvura | DMSO: 20MG / ML |
Viagra, sildenafil citrate; 1 - [[3- (4,7-Dihydro-1-methyl-7-quyl-3h-pyrazolo [4-d) -4-ethoxyphene] -4-methylpisekuva 5 - 1 - [[3- (6,7-Dihydro-1-methyl-7-proyl-1h-pyrichalo [4-d)-ethylpheerl] -4-methylpemErazine, 2-hydroxy-1,2,3-pranetricarboylate; Sildenafilcitrate (100mg); Sildenafilcrate,> = 99%; svibisafirate, nyanzvi. 5- [2-ethoxy-5 - [(4-methyl-piperazin-1-yl) sulfonyl] phenyl]-1-methyl-3h-pyrazolo
Pharmacological chiito
Sildenafil Citrate is sarudza 5-phosphodieseralserse inhibitor nitric n oxidesphate Pamusoro pekuwedzera kwakananga kwemidziyo yeropa yeropa, inogona zvakare kudzivirira kana kudzosera kumashure kwekugadzirisa.
Mishonga yemishonga uye zvikumbiro
Sildengil Citrate, Trade zita Viagre, inowanzozivikanwa seViagra, is cyclic guanosphate (CGMP) Sildenafil Citrate inogona kusimudzira mhedzisiro yeNitric oxide (no) nekudzora iyo Type 5 phosphodieserese cyclic guanosphate (cgm) muCorpus Cavernosum. Wedzera mwero weCGMP muCorpus Cavernosum, zorora tsandanyama yeCorpus muCorpus Cavernosum, wedzera kupenya kweropa, kuwedzera iyo penis eered nguva uye kuwedzera kusimba. Kune varwere vasina kusimba vane erectile dysfunction. Vakuru vanotora makumi mashanu emuromo nomuromo mumwe nemumwe, kusvika 1 nguva pazuva, uye shandisa sezvazvinodiwa dzinenge 1 awa isati yasvika pabonde. Mari yakakwira ndeye 0.1g nguva imwe neimwe.
MuVivo Zvidzidzo
Imbwa dzinonakidza, sildengil citrate inosimudzira penile eerectile service pasi pelvic nerve kukurudzira nekuyera kumanikidza intracaravaraveronous. Sildengil citrate zvakachinja zvakarongedzwa zvisina kujairika carbamoylcholine-yakakurudzirwa zororo uye yakadzivirirwa superoxide kuumbwa mune cavernosal tishu yehypercholestelestecemic Mune Sprague-Dawley makonzo, Sildengil inovandudza erectile basa mune imwe nzira-inoenderana-inoenderana, nekuwedzera kwekupora kuri kuitika pazuva 28 pane dofo ye20 mg / kg pazuva. Mune Sprague-Dawley makonzo, kutonga kweSildenfil kwakaguma neakatsetseka yemaswiyo yeColagen yeColagen yekuchengetedza uye kuchengetedzwa kweCD31 uye Enos kutaura. Mune Sprague makonzo, Sildenfil zvakanyanya kuderedza indekisi yeapopotic uye yakawedzera pophorylation ye AKT uye Enosi kana achienzaniswa neboka rekutonga.