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Sildenafil Citrate kurapa erectile dysfunction 171599-83-0

Tsananguro pfupi:

Chemical formula: c28h38n6o11s

Sollear Huremu: 666.70

Cas nhamba: 171599-83-0

Einecs nhamba: 200-659-6

Inline Pfungwa: 187-189 ℃

Boling Point: 672.4 ℃

Flash Point: 360.5 ℃

Density: 1.445g / cm3

Refractive Index: 1.683


Chigadzirwa Chinhu

Zvigadzirwa tags

Chigadzirwa Chinhu

Zita Sildenafil Citrate
Nhamba 171599-83-0
Molecular Formula C28h38n6o11s
Sreek inoremerwa 666.70
Einecs nhamba 200-659-6
Merck 14,8489
Density 1.445G / cm3
Kuchengetedza mamiriro 2-8 ° C
Fomu Poda
Ruvara Chena
Solubility yemvura DMSO: 20MG / ML

Synonyms

Viagra, sildenafil citrate; 1 - [[3- (4,7-Dihydro-1-methyl-7-quyl-3h-pyrazolo [4-d) -4-ethoxyphene] -4-methylpisekuva 5 - 1 - [[3- (6,7-Dihydro-1-methyl-7-proyl-1h-pyrichalo [4-d)-ethylpheerl] -4-methylpemErazine, 2-hydroxy-1,2,3-pranetricarboylate; Sildenafilcitrate (100mg); Sildenafilcrate,> = 99%; svibisafirate, nyanzvi. 5- [2-ethoxy-5 - [(4-methyl-piperazin-1-yl) sulfonyl] phenyl]-1-methyl-3h-pyrazolo

Pharmacological mhedzisiro

Pharmacological chiito
Sildenafil Citrate is sarudza 5-phosphodieseralserse inhibitor nitric n oxidesphate Pamusoro pekuwedzera kwakananga kwemidziyo yeropa yeropa, inogona zvakare kudzivirira kana kudzosera kumashure kwekugadzirisa.

 

Mishonga yemishonga uye zvikumbiro
Sildengil Citrate, Trade zita Viagre, inowanzozivikanwa seViagra, is cyclic guanosphate (CGMP) Sildenafil Citrate inogona kusimudzira mhedzisiro yeNitric oxide (no) nekudzora iyo Type 5 phosphodieserese cyclic guanosphate (cgm) muCorpus Cavernosum. Wedzera mwero weCGMP muCorpus Cavernosum, zorora tsandanyama yeCorpus muCorpus Cavernosum, wedzera kupenya kweropa, kuwedzera iyo penis eered nguva uye kuwedzera kusimba. Kune varwere vasina kusimba vane erectile dysfunction. Vakuru vanotora makumi mashanu emuromo nomuromo mumwe nemumwe, kusvika 1 nguva pazuva, uye shandisa sezvazvinodiwa dzinenge 1 awa isati yasvika pabonde. Mari yakakwira ndeye 0.1g nguva imwe neimwe.

 

MuVivo Zvidzidzo
Imbwa dzinonakidza, sildengil citrate inosimudzira penile eerectile service pasi pelvic nerve kukurudzira nekuyera kumanikidza intracaravaraveronous. Sildengil citrate zvakachinja zvakarongedzwa zvisina kujairika carbamoylcholine-yakakurudzirwa zororo uye yakadzivirirwa superoxide kuumbwa mune cavernosal tishu yehypercholestelestecemic Mune Sprague-Dawley makonzo, Sildengil inovandudza erectile basa mune imwe nzira-inoenderana-inoenderana, nekuwedzera kwekupora kuri kuitika pazuva 28 pane dofo ye20 mg / kg pazuva. Mune Sprague-Dawley makonzo, kutonga kweSildenfil kwakaguma neakatsetseka yemaswiyo yeColagen yeColagen yekuchengetedza uye kuchengetedzwa kweCD31 uye Enos kutaura. Mune Sprague makonzo, Sildenfil zvakanyanya kuderedza indekisi yeapopotic uye yakawedzera pophorylation ye AKT uye Enosi kana achienzaniswa neboka rekutonga.

 

 


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