Zita | Desmopressin |
CAS nhamba | 16679-58-6 |
Molecular formula | C46H64N14O12S2 |
Molecular uremu | 1069.22 |
Nhamba yeEINECS | 240-726-7 |
Kutenderera chaiko | D25 +85.5 ± 2 ° (yakaverengerwa peptide yemahara) |
Density | 1.56±0.1 g/cm3(Zvakafanotaurwa) |
RTECS Nha. | YW9000000 |
Kuchengetedza mamiriro | Chengeta pa 0°C |
Solubility | H2O: soluble20mg/mL, yakajeka, isina ruvara |
Acidity coefficient | (pKa) 9.90±0.15 (Zvakafanotaurwa) |
MPR-TYR-PHE-GLN-ASN-CYS-PRO-D-ARG-GLY-NH2;MINIRIN;[DEAMINO1, DARG8] VASOPRESSIN;[DEAMINO-CYS1, D-ARG8]-VASOPRESSIN;DDAVP, MUNHU;DESMOPRESSIN;DESMOPRESSIN, MUNHU;DESAMINO-[D-ARG8] VASOPRESSIN
(1) Kurapa kwepakati chirwere cheshuga insipidus.Mushure memushonga unogona kuderedza urinary excretion, kuderedza weti frequency uye kuderedza nocturia.
(2) Kurapa kweusiku enuresis (varwere vane makore 5 kana kupfuura).
(3) Edza renal weti yekutarisa basa, uye ita mutsauko wekuongororwa kwe renal basa.
(4) Kune hemophilia nezvimwe zvirwere zvekubuda ropa, chigadzirwa ichi chinogona kupfupisa nguva yekubuda ropa uye kudzivirira kubuda ropa.Inogona kuderedza kuwanda kwekurasikirwa kweropa kwemukati uye postoperative oozing;kunyanya pamwe chete nekudzikama kunodzorwa kweropa panguva yekuvhiyiwa, inogona kuderedza kubuda kweropa kubva kune nzira dzakasiyana-siyana, uye kuderedza kubuda kwemashure, izvo zvinogona kuita basa rakanaka mukudzivirira ropa.
Chirwere cheshuga insipidus chinonyanya kukanganisa kwemetabolism yemvura inoratidzirwa nekuwanda weti kubuda, polydipsia, hypoosmolarity, uye hypernatremia.Kusakwana kana kukwana kwevasopressin (central diabetes insipidus), kana renal insufficiency yevasopressin (nephrogenic diabetes insipidus) inogona kutanga.Kliniki, chirwere cheshuga insipidus chakafanana neprimary polydipsia, mamiriro ezvinhu umo kunwa mvura yakawandisa kunokonzerwa nekusashanda zvakanaka kwemaitiro ekudzora kana nyota isina kujairika.Kusiyana neprimary polydipsia, kuwedzera kwekudya kwemvura kune varwere vane chirwere cheshuga insipidus inoenderana nekuchinja kweosmotic pressure kana ropa.