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Linaclotide yeGastrointestinal Disorders 851199-59-2

Tsanangudzo Pfupi

Zita: Linaclotide

Nhamba yeCAS: 851199-59-2

Molecular formula: C59H79N15O21S6

Molecular uremu: 1526.74


Product Detail

Product Tags

Product Detail

Zita Linaclotide
CAS nhamba 851199-59-2
Molecular formula C59H79N15O21S6
Molecular uremu 1526.74

Mashoko anoreva zvakafanana

Linacllotide;Linaclotide;LinaelotideAcetate;Linaelotide;CY-14;Liclotide;Argpessin;L-Tyrosine,L-cysteineyl-L-cysteineyl-L-α-glutamyl-L-tyrosyl-L-cysteinyl-L-cysteinyl-L-asparaginyl- L-prolyl-L-alanyl-L-cysteineyl-L-threonylglycyl-L-cysteineyl-,cyclic(1→6),(2→10),(5→13)-tris(disulfide)

Tsanangudzo

Linaclotide, yakagadzirwa peptide chimiro ine gumi nemana amino acids, ine hukama nemhuri inogadzika guanosine peptide uye ndiyo yega FDA-inotenderwa GC-C (guanylate) Cyclase-C) agonist mishonga yekurapa irritable bowel syndrome nekuzvimba (IBS- C) uye chisingaperi idiopathic constipation (CIC) muvakuru.

Chemical Properties

Linaclotide ichena kusvika kune-white amorphous powder;zvishoma soluble mumvura uye aqueous sodium chloride mhinduro (0.9%).

Zvinoshanda sei

Linaclotide inonzi guanylate cyclase-C receptor agonist (GCCA) ine zvose visceral analgesic uye endocrine basa.Zvose linaclotide uye metabolite yayo inoshanda inogona kusunga kune guanylate cyclase-C (GC-C) receptor pane luminal pamusoro peiyo diki intestinal epithelium.Mune mhando dzemhuka, linaclotide inoderedza marwadzo evisceral uye inowedzera gastrointestinal kufambisa kuburikidza nekuita kweGC-C, uye muvanhu, mushonga unowedzerawo colonic transit.Mhedzisiro yeGC-C activation yakawedzera intracellular uye extracellular cGMP (cyclic guanosine monophosphate) concentrations.Extracellular cGMP inogona kuderedza kuita kwemarwadzo tsinga fibers uye kuderedza visceral kurwadziwa mumuenzaniso mhuka.Intracellular cGMP inogona kuwedzera secretion yekloridi uye bicarbonate mudumbu diki nekuita CFTR (cystic fibrosis transmembrane conductance regulator), iyo inozopedzisira yaita kuti kuwedzerwa kwemukati memukati memukati mese uye nekumhanya kwediki intestinal transit.

FAQ

Iwe unovimbisa zvakachengeteka uye zvakachengeteka kuendesa zvigadzirwa?

Ehe, isu tinogara tichishandisa emhando yepamusoro ekunze kurongedza.Isu tinoshandisawo yakasarudzika njodzi yekurongedza kune zvinhu zvine njodzi uye yakatenderwa inotonhora yekuchengetedza inotakura kune tembiricha zvinhu.Nyanzvi kurongedza uye zvisiri-yakajairwa kurongedza zvinodiwa zvinogona kuunza imwe mari.

Zvakadini nemari yekutumira?

Mutengo wekutumira unoenderana nenzira yaunosarudza kuwana zvinhu.Express ndiyo nzira inokurumidza asi zvakare inodhura zvakanyanya.Nekutakura zvinhu mugungwa ndiyo yakanakisa mhinduro kune yakakura mari.Chaiyo mitengo yekutakura tinogona kukupa chete kana tichiziva ruzivo rwehuwandu, huremu uye nzira.Ndapota taura nesu kuti uwane rumwe ruzivo.


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