Zita | CARBETOCIN |
CAS nhamba | 37025-55-1 |
Molecular formula | C45H69N11O12S |
Molecular uremu | 988.17 |
Nhamba yeEINECS | 253-312-6 |
Kutenderera chaiko | D -69.0° (c = 0.25 mu1M acetic acid) |
Boiling point | 1477.9±65.0 °C (Zvakafanotaurwa) |
Density | 1.218±0.06 g/cm3(Zvakafanotaurwa) |
Kuchengetedza mamiriro | -15°C |
Form | upfu |
BUTYRYL-TYR(ME)-ILE-GLN-ASN-CYS-PRO-LEU-GLY-NH2, (SULFIDEBODBETWEENBUTYL-4-YLANDCYS);BUTYRYL-TYR(ME)-ILE-GLN-ASN-CYS-PRO-LEU-GLY-NH2TRIFLUOROACETATESALT;(BUTYRYL1, TYR(ME)2)-1-CARBAOXYTOC INTRIFLUOROACETATESALT;(BUTYRYL1, TYR(ME)2)-OXYTOCIN;(BUTYRYL1,TYR(ME)2)-OXYTOCINTRIFLUOROACETATESALT;CARBETOCIN;CARBETOCINTRIFLUOROACETATESALT;(2-O-METHYLTYROSINE)-DE-AMINO-1-CARBAOXYTOCIN
Carbetocin, an oxytocin (OT) analog, inonzi oxytocin receptor agonist ine Ki ye7.1 nM.Carbetocin ine hukama hwepamusoro (Ki = 1.17 μM) ye chimeric N-terminus ye oxytocin receptor.Carbetocin ine mukana wekutsvaga kwekubuda kweropa mushure mekusununguka.Carbetocin inogona kupinda mukati meropa-brain barriers uye ine antidepressant-sekuita sekuita nekuita oxytocin receptors muCNS.
Carbetocin is a synthetic long-acting oxytocin 8-peptide analog ine agonist properties, uye maitiro ayo ekiriniki uye pharmacological akafanana neaya anongoitika oxytocin.Senge oxytocin, carbetocin inosunga kune mahormone receptors euterine yakatsetseka tsandanyama, zvichikonzera rhythmic contractions yechibereko, ichiwedzera kuwanda kwayo uye kuwedzera uterine toni pahwaro hwekumanikana kwepakutanga.Oxytocin receptor mazinga muchibereko akaderera mumamiriro asina pamuviri, anowedzera panguva yekuzvitakura, uye peak panguva yekusununguka.Nokudaro, carbetocin haina simba kune chibereko chisina pamuviri, asi ine simba rakasimba rekuita chibvumirano pamimba ine pamuviri uye ichangobva kugadzirwa.
Shanduko dzinodzorwa zvinoenderana nemaitiro.Zvichienderana nemhedzisiro uye njodzi uye kuomarara, shanduko dzinoiswa seMakuru, Diki uye Saiti.Shanduko dzesaiti dzine zvishoma pakuchengetedza uye kunaka kwechigadzirwa, uye saka hazvidi kubvumidzwa uye chiziviso kune mutengi;Shanduko diki dzine mhedzisiro ine pakati pekuchengetedza uye kunaka kwechigadzirwa, uye inoda kuzivisa mutengi;Shanduko huru dzine mhedzisiro yepamusoro pakuchengetedza uye kunaka kwechigadzirwa, uye inoda kubvumidzwa nemutengi.
Zvinoenderana nemaitiro, shanduko yekutonga inotangwa neshanduko application umo shanduko yeruzivo uye zvine musoro kune shanduko inotsanangurwa.Ongororo yacho inozoitwa zvichitevera chikumbiro, icho chinoitwa nekuchinja kutonga kwakakodzera madhipatimendi.Zvichakadaro, iyo shanduko yekutonga inokamurwa kuita Major level, General level uye Diki level.Mushure mekuongorora kwakakodzera pamwe nekuiswa, ese nhanho shanduko yekutonga inofanirwa kubvumidzwa neQA Manager.Iyo shanduko yekutonga inoitwa mushure mekubvumidzwa zvinoenderana nehurongwa hwekuita.Iyo shanduko yekutonga inozovharwa mushure mekunge QA yasimbisa shanduko yekutonga yaitwa nemazvo.Kana ichibatanidza chiziviso chemutengi, mutengi anofanira kuziviswa nenguva mushure mekuchinja shanduko kubvumidzwa